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Tirzepatide exhibits a prolonged circulating half-life of approximately 120150 hours, enabling sustained receptor engagement [3]

Targeting mitochondrial quality control for diabetic cardiomyopathy: Therapeutic potential of hypoglycemic drugs

10.1016/j.molmet.2020.101102 34 PatouliasD.StavropoulosK.ImprialosK.KatsimardouA.KalogirouM

doi: 10.1002/dmrr.3070 [DOI] [PubMed] [Google Scholar] 61.Cirincione B, Mager DE

Remarkably, G49-mediated beiging was blocked by GCGRant or Atglistatin that, in addition to lipolysis, also suppressed the increase in Ucp1 expression in eWAT, again linking lipolysis with eWAT browning
